måndag 8 december 2014

A giant leap for drug delivery (also vaccines)


Highly Stable Formulation of Any Compounds with Differential Solubility

NOVEL SOLID INEXPENSIVE FORMULATION IN A MAGNESIUM CAPSULE





CHALLENGE

Copy of seeker summary from the Innocentive Webb site:


DISCLAIMERS
  • THIS IS A STUB SOLUTION TO BE EXPANDED
  • IP DISCLAIMER, THE IP TRANSFER FOR THIS SOLUTION WILL BE ONLY FOR THE PROPOSED COMPOUNDS, NOT FOR OTHER CHEMICAL ENTITIES, A LICENSING AGREEMENT IS ALSO AN OPTION
  • WE ALSO HAVE A VERSION OF THE CAPSULE THAT IS A ONCE-A-WEEK INJECTION WITH TIMED “INJECTIONS/DISSOLVEMENT” OF ONE DOSE A DAY FOR ONE WEEK. THIS SOLUTION IS HOWEVER NOT INCLUDED IN THE SOLUTION OR THE IP TRANSFERRED AND IS ONLY COMMUNICATED FOR INFORMATION PURPOSES
  • AND A  LICENSING AGREEMENT COULD BE ADVANTAGEOUS TO BOTH PARTIES A LONG THE LINES OF WHAT IS MENTIONED IN THE PROBLEM DESCRIPTION

WHAT IS THE PROPOSED SOLUTION?


  • THE SOLUTION IS A SOLID FORMULATION THAT WE HAVE A LOT OF EXPERIENCE WITH
  • IT CONSISTS OF THE TWO COMPOUNDS ENCAPSULATED IN A SOLID CAPSULE OF PURE MAGNESIUM
  • THE CAPSULE CAN BE QUICKLY AND SAFELY INJECTED INTRA-MUSCULAR AND SUB-CUTANEOUS IN ANY ANIMAL
  • INJECTION IS DONE THOUGH A NORMAL NEEDLE WITH 1,5 MM INNER DIAMETER
  • THE MAGNESIUM WILL BIO-CORRODE WITHIN MINUTES IN BODILY FLUIDS
  • AND THE TWO COMPOUNDS WILL BE DISSOLVED QUICKLY IN BODILY FLUIDS
  • ACCORDING TO OUR CALCULATIONS THE PROPERTIES OF THE TWO COMPOUNDS ARE SUITABLE FOR THIS METHOD, RESULTING IN A FEW MILLIMETER LONG MAGNESIUM CAPSULE
  • THE DRY SUBSTANCE MAGNESIUM ENCAPSULATED CAPSULE IS PRE-LOADED INTO AN INEXPENSIVE NEEDLE WITH PLASTICS HOLDER FOR INJECTION, THE SAME AS DEVICE OFTEN OFTEN USED FOR MARKING OF ANIMALS WITH RFID-TAGS
  • IN RARE CASES THE MAGNESIUM CAPSULE HAS A THIRD COMPARTMENT WITH A SOLVENT, BUT WE DO NOT JUDGE THAT AS NECESSARY IN THIS CASE
  • SHELF-LIFE IS ALMOST UN-LIMITED IN SOLID FORM AN INERT ATMOSPHERE INSIDE THE MAGNESIUM CAPSULE
  • THE STERILE PRE-PACKED “SYRINGE” IS NOT SENSITIVE TO HUMIDITY
  • THE TECHNOLOGY ALLOWS FOR VERY INEXPENSIVE MANUFACTURING
  • THE TWO COMPOUNDS ARE KEPT APART IN DIFFERENT COMPARTMENTS IN THE CAPSULE AND DO NOT AFFECT EACH OTHER DURING STORAGE
  • THE DISSOLVED MAGNESIUM IS POSITIVE FOR THE ORGANSISM

  • AVERAGE COST OF GOODS IN MASS PRODUCTION FOR THE DRUG DELIVERY TECHNIQUE IS A FEW CENTS.
  • WE ALSO HAVE A VERSION OF THE CAPSULE THAT IS A ONCE-A-WEEK INJECTION WITH TIMED “INJECTIONS/DIS-SOLVEMENT” OF ONE DOSE A DAY FOR ONE WEEK. THIS SOLUTION IS HOWEVER NOT INCLUDED IN THE SOLUTION OR THE IP TRANSFERRED AND IS ONLY COMMUNICATED FOR INFORMATION PURPOSES. THERE IS ALSO A COMPUTER CONTROLLED VERSION THAT CAN HANDLE COMPLEX DOSING SCHEMES, BUT THAT SOLUTION REQUIRES EXPLANTATION AFTER ALL DOSES ARE GIVEN.

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